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Tepotinib chemical structure

Tepotinib

Regular price $148.00 USD
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THE SCIENCE, IN DETAIL

Know your product.

Specifications
Big target
Protein Tyrosine Kinase
Cas number
1100598-32-0
Formula
C29H28N6O2
Small target
c-Met
Smiles
CN1CCC(CC1)COC2=CN=C(N=C2)C3=CC=CC(=C3)CN4C(=O)C=CC(=N4)C5=CC=CC(=C5)C#N
Storage conditions
2 years -80 in solvent
Synonyms
EMD 1214063, MSC2156119
Scientific background
Tepotinib is a potent and selective c-Met inhibitor with IC50 of 4 nM, >200-fold selective for c-Met than IRAK4, TrkA, Axl, IRAK1, and Mer. Tepotinib (EMD 1214063) induces autophagy. Phase 1.
Technical documents

Documents

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