Pelabresib (CPI-0610)

Name: Pelabresib (CPI-0610)
Brand: Selleckchem
Price: 224.0 USD
Availability: InStock

Vendor: Selleckchem

Type: Epigenetics

SKU: S7853-5mg

$224.00 USD

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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Big target

Epigenetics

Cas number

1380087-89-7

Formula

C20H16ClN3O2

Small target

Epigenetic Reader Domain

Smiles

CC1=NOC2=C1C3=CC=CC=C3C(=NC2CC(=O)N)C4=CC=C(C=C4)Cl

Storage conditions

2 years -80 in solvent

Background

Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.

Pelabresib (CPI-0610)

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Product Overview

Background

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