APS-2-79 HCl chemical structure

APS-2-79 HCl

Vendor: Selleckchem

Type: Protein Tyrosine Kinase

SKU: S8355-5mg

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APS-2-79 HCl chemical structure

APS-2-79 HCl

$110.00 USD

THE SCIENCE, IN DETAIL

Know your product.

Specifications
Big target
Protein Tyrosine Kinase
Cas number
2002381-31-7
Formula
C23H21N3O3.HCl
Small target
MEK
Smiles
CC1=C(C=CC(=C1)OC2=CC=CC=C2)NC3=NC=NC4=CC(=C(C=C43)OC)OC.Cl
Storage conditions
2 years -80 in solvent
Scientific background
APS-2-79 is a MAPK antagonist that modulating KSR-dependent MAPK signalling by antagonizing RAF heterodimerization as well as the conformational changes required for phosphorylation and activation of KSR-bound MEK. IC50=120 ± 23 nM.
Technical documents

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