Padnarsertib (KPT 9274) chemical structure

Padnarsertib (KPT 9274)

Vendor: Selleckchem

Type: Metabolism

SKU: S8444-2mg

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Padnarsertib (KPT 9274) chemical structure

Padnarsertib (KPT 9274)

$110.00 USD

THE SCIENCE, IN DETAIL

Know your product.

Specifications
Big target
Metabolism
Cas number
1643913-93-2
Formula
C35H29F3N4O3
Small target
NAMPT
Smiles
C1CN(CCC1(F)F)C(=O)C2=CC=C(C=C2)C3=CC(=C4C(=C3)C=C(O4)CNC(=O)C=CC5=CN=C(C=C5)N)C6=CC=C(C=C6)F
Storage conditions
2 years -80 in solvent
Scientific background
Padnarsertib (KPT 9274) is an orally bioavailable small molecule that is a non-competitive dual inhibitor of PAK4 and NAMPT. It shows an IC50 of ~120 nM for NAMPT in a cell-free enzymatic assay.
Technical documents

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