Selpercatinib (LOXO-292)

Vendor: Abmole

Type: Molecular

SKU: M9900

$92.00 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Selpercatinib (LOXO-292) is a first-in-class, highly selective and potent small molecule RET inhibitor with good blood-brain barrier (BBB) penetration. and RET (G810R) with IC50 values of 14.0 nM, 24.1 nM and 530.7 nM, respectively.
Casnumber
2152628-33-4
Formula
C29H31N7O3
Mw
525.6
Psmiles
COC1=NC=C(CN2C3CC2CN(C3)C4=NC=C(C=C4)C5=CC(=C[N]6N=CC(=C56)C#N)OCC(C)(C)O)C=C1
Purity
99.98%
Solubility
DMSO 20 mg/mL
Target synonyms
LOXO-292; ARRY-192
Selpercatinib (LOXO-292)

Selpercatinib (LOXO-292)

$92.00 USD