Serabelisib

Vendor: Abmole

Type: Molecular

SKU: M6175

$166.75 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Serabelisib (INK-1117,MLN-1117,TAK-117) is a potent and selective oral PI3Kα isoform inhibitor (IC50 of 21 nmol/L against PI3Kα) that has demonstrated > 100-fold selectivity relative to other class I PI3K family members (PI3Kβ/γ/δ) and mTOR, and a high degree of selectivity against many other kinase.
Casnumber
1268454-23-4
Formula
C19H17N5O3
Mw
363.37
Psmiles
NC1=NC2=C(O1)C=CC(=C2)C3=C[N]4C(=NC=C4C(=O)N5CCOCC5)C=C3
Purity
>99.0%
Solubility
16 mg/mL in DMSO
Target synonyms
INK-1117,MLN-1117,TAK-117
Serabelisib

Serabelisib

$166.75 USD