Sparsentan (RE-021)

Vendor: Abmole

Type: Molecular

SKU: M20689

$120.75 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Sparsentan (PS-433540, RE-021, DARA) is a first-in-class, orally active, high-affinity dual antagonist of the endothelin type A receptor (ETA) and Angiotensin II type 1 (AT1) receptor, with Ki values of 9.3 and 0.8 nM, respectively.
Casnumber
254740-64-2
Formula
C32H40N4O5S
Mw
592.75
Psmiles
CCCCC1=NC2(CCCC2)C(=O)N1CC3=CC=C(C(=C3)COCC)C4=CC=CC=C4[S](=O)(=O)NC5=NOC(=C5C)C
Purity
>99%
Solubility
DMSO 90 mg/mL
Target synonyms
PS-433540; RE-021; DARA-a; BMS-346567
Sparsentan (RE-021)

Sparsentan (RE-021)

$120.75 USD