Tenalisib

Vendor: Abmole

Type: Molecular

SKU: M7538

$149.50 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Tenalisib (RP6530) is a potent and selective dual PI3Kδ/γ inhibitor with IC50 values of 24.5 nM and 33.2 nM for PI3Kδ and PI3Kγ, respectively. Its selectivity over α and β isoforms are more than 300-fold and 100-fold, respectively.
Casnumber
1639417-53-0
Formula
C23H18FN5O2
Mw
415.42
Psmiles
CCC(NC1=C2N=C[NH]C2=NC=N1)C3=C(C(=O)C4=CC=CC=C4O3)C5=CC=CC(=C5)F
Purity
>98.0%
Solubility
75 mg/mL in DMSO
Target synonyms
RP6530
Tenalisib

Tenalisib

$149.50 USD