THIP hydrochloride

Vendor: Abmole

Type: Molecular

SKU: M7410

$195.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
THIP hydrochloride (Gaboxadol hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 μM). Gaboxadol hydrochloride displays a partial agonist efficacy on subunit α1β2γ2 with an ED50 value of 143 µM, a full agonist efficacy at α5 subunit (ED50=28-129 µM) and a superagonist efficacy at α4β3δ (ED50=6 µM).
Casnumber
85118-33-8
Formula
C6H8N2O2.HCl
Mw
176.6
Psmiles
C1CNCC2=C1C(=O)NO2.Cl
Purity
>99.0%
Solubility
DMSO 17.66 mg/mL
Target synonyms
Gaboxadol hydrochloride; Lu 02-030 HCl
THIP hydrochloride

THIP hydrochloride

$195.50 USD