THZ2

Vendor: Abmole

Type: Molecular

SKU: M8995

$345.00 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
THZ2 (an analog of THZ1) is a potent and selective CDK7 inhibitor which overcomes the instability of THZ1 in vivo (IC50s: CDK7=13.9 nM; TNBC cells=10 nM).
Casnumber
1604810-84-5
Formula
C31H28ClN7O2
Mw
566.05
Psmiles
CN(C)C\C=C\C(=O)NC1=CC=CC(=C1)C(=O)NC2=CC=CC(=C2)NC3=NC=C(Cl)C(=N3)C4=C[NH]C5=CC=CC=C45
Purity
>99.0%
Solubility
DMSO: ≥ 30 mg/mL
THZ2

THZ2

$345.00 USD