Tolinapant(ASTX660)

Vendor: Abmole

Type: Molecular

SKU: M9933

$310.50 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
ASTX660 is a potent, non-peptidomimetic antagonist of cIAP1/2 and XIAP, it potently inhibited the interactions between a SMAC-derived peptide and the BIR3 domains of XIAP (BIR3-XIAP) and cIAP1 (BIR3-cIAP1) with IC50 values less than 40 and 12 nmol/L, respectively.
Casnumber
1799328-86-1
Formula
C30H42FN5O3
Mw
539.68
Psmiles
CC1CN(CC(=O)N2CC(C)(C)C3=C2C=C(CC4=CC=C(F)C=C4)C(=N3)CO)C(CN1)CN5CCOCC5C
Purity
>98%
Solubility
DMSO ≥ 80 mg/mL
Target synonyms
ASTX-660
Tolinapant(ASTX660)

Tolinapant(ASTX660)

$310.50 USD