Umbralisib

Vendor: Abmole

Type: Molecular

SKU: M5268

$235.75 USD
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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Umbralisib (TGR-1202) is an orally active, potent and selective dual PI3Kδ and casein kinase-1-ε (CK1ε) inhibitor, with EC50 of 22.2 nM and 6.0 μM, respectively.
Casnumber
1532533-67-7
Formula
C31H24F3N5O3
Mw
571.55
Psmiles
CC(C)OC1=C(F)C=C(C=C1)C2=N[N](C(C)C3=C(C4=CC(=CC=C4)F)C(=O)C5=CC(=CC=C5O3)F)C6=C2C(=NC=N6)N
Purity
>98.5%
Solubility
DMSO 25 mg/mL
Target synonyms
TGR-1202; RP5264
Umbralisib

Umbralisib

$235.75 USD