Varenicline dihydrochloride

Vendor: Abmole

Type: Molecular

SKU: M20984

$149.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
Varenicline (CP 526555, Chantix, Champix) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation.
Casnumber
866823-63-4
Formula
C13H15Cl2N3
Mw
284.18
Psmiles
Cl.Cl.C1NCC2CC1C3=CC4=NC=CN=C4C=C23
Purity
>99%
Solubility
DMSO 57 mg/mL; Water 57 mg/mL
Target synonyms
Chantix, Champix
Varenicline dihydrochloride

Varenicline dihydrochloride

$149.50 USD