VER-246608

Vendor: Abmole

Type: Molecular

SKU: M28806

$241.50 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
VER-246608 is a potent and ATP-competitive inhibitor of pyruvate dehydrogenase kinase (PDK) with IC50s of 35 nM, 40 nM, 84 nM, and 91 nM for PDK-1, PDK-3, PDK-2, and PDK-4, respectively.
Casnumber
1684386-71-7
Formula
C28H23ClF2N4O4
Mw
552.96
Psmiles
CC1=CN=C(N=C1C2=CC=C(C=C2)N(CC3=CC=C(C=C3)CNC(=O)C(F)F)C(=O)C4=C(C=C(C=C4)O)O)Cl
Purity
≥98.5%
Solubility
DMSO 100 mg/mL (ultrasonic)
VER-246608

VER-246608

$241.50 USD