VU0467154

Vendor: Abmole

Type: Molecular

SKU: M28478

$201.25 USD
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Available in stock (500)

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For research use only — not intended for clinical or diagnostic purposes.

Product Overview

Bioactivity
VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor (mAChR), potentiating the response to ACh with pEC50s of 7.75, 6.2 and 6 for rat, human and cynomolgus monkey M4 receptor, respectively.
Casnumber
1451993-15-9
Formula
C17H15F3N4O3S2
Mw
444.45
Psmiles
CC1=C(N=NC2=C1C(=C(S2)C(=O)NCC3=CC=C(C=C3)S(=O)(=O)C(F)(F)F)N)C
Purity
≥99.0%
Solubility
DMSO 13.89 mg/mL (ultrasonic)
VU0467154

VU0467154

$201.25 USD