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Zamicastat

Zamicastat

Regular price $569.25 USD
Sale price Regular price

THE SCIENCE, IN DETAIL

Know your product.

Specifications
Bioactivity
Zamicastat is a dopamine β-hydroxylase (DBH) inhibitor that crosses the blood-brain barrier and causes central and peripheral effects. In addition, Zamicastat is a concentration-dependent dual P-gp and BCRP inhibitor with IC50 values of 73.8 μM and 17.0 μM, respectively.
Casnumber
1080028-80-3
Formula
C21H21F2N3OS
Mw
401.47
Psmiles
C1C(COC2=C1C=C(C=C2F)F)N3C(=CNC3=S)CCNCC4=CC=CC=C4
Purity
>98.0%
Solubility
DMSO >100 mg/mL
Target synonyms
BIA 5-1058
Technical documents

Documents

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