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Zetomipzomib maleate

Zetomipzomib maleate

Regular price $3,277.50 USD
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THE SCIENCE, IN DETAIL

Know your product.

Specifications
Bioactivity
Zetomipzomib (KZR-616) maleate is a first-in-class inhibitor of immunoproteasome that selectively targets the immunoproteasome subunit LMP7 (IC50: 39/57 nM=hLMP7/mLMP7) and LMP2 (IC50:131/179 nM=hLMP7/mLMP7). Potential of Zetomipzomib maleate for use in multiple autoimmune diseases.
Casnumber
2170983-62-5
Formula
C34H46N4O12
Mw
702.75
Psmiles
CC(C(=O)NC(C(C1=CC=C(C=C1)OC)O)C(=O)NC(CC2=CCCC2)C(=O)C3(CO3)C)NC(=O)CN4CCOCC4.C(=CC(=O)O)C(=O)O
Purity
>99%
Solubility
DMSO ≥ 200 mg/mL
Target synonyms
KZR-616 maleate
Technical documents

Documents

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